1. 100 Years of the Biginelli Dihydropyrimidine Synthesis.
C.O. Kappe
Tetrahedron 1993, 49, 6937-6963 (Tetrahedron Report Number 336).
2. The Use of 1,2-Shifts in Carbenes and Nitrenes in the Generation of Novel Heterocumulenes.
C. Wentrup, C.O. Kappe, M.W. Wong
Pure Appl. Chem. 1995, 67, 749-754.
3. Synthetic Applications of Furan Diels-Alder Chemistry
C.O. Kappe, S. Murphree, A. Padwa
Tetrahedron 1997, 53, 14179-14233 (Tetrahedron Report Number 430)
4. 4-Aryldihydropyrimidines via the Biginelli Condensation: Aza-Analogs of Niffedipine-Type Calcium Channel Modulators.
C.O. Kappe
Molecules 1998, 3, 1-9.
5. Perfluorinated Acyl(Aroyl)pyruvates as Building Blocks for the Synthesis of Heterocycles.
V.I. Saloutin, Y.U. Burgart, C.O. Kappe, O.N. Chupakhin
Heterocycles 2000, 52, 1411-1434.
6. Recent Advances in the Biginelli Dihydropyrimidine Synthesis. New Tricks from an Old Dog.
C.O. Kappe
Acc. Chem. Res. 2000, 33, 879-888.
7. Biologically Active Dihydripyrimidones of the Bignelli-Type. A Literature Survey.
C.O. Kappe
Eur. J. Med. Chem. 2000, 35, 1043-1052.
8. Speeding Up Solid-Phase Chemistry by Microwave Irradiation. A New Tool for High-Throughput Synthesis.
C.O. Kappe
American Laboratory 2001, 33(10), 13-19.
9. On the Chemistry of Stable a-Oxoketenes.
G. Kolenz, W. Heilmayer, C.O. Kappe, B. Wallfish, C. Wentrup
Croat. Chim. Acta 2001, 74, 815-823.
10. High-Speed Combinatorial Synthetics Utilizing Microwave Irradiation.
C.O. Kappe
Curr. Opin. Chem. Biol. 2002, 6, 314-320.
11. The Generation of Dihydropyrimidine Libraries Utilizing Biginelli Multicomponent Chemistry.
C.O. Kappe
QSAR Comb. Sci. 2003, 22, 630-645.
12. Solid- and Solution-Phase Synthesis of Bioactive Dihydropyrimidines.
D. Dallinger, A. Stadler, C.O. Kappe
Pure Appl. Chem. 2004, 76, 1017-1024.
13. Controlled Microwave Heating in Modern Organic Synthesis.
C.O. Kappe
Angew. Chem. Int. Ed. 2004, 43, 6250-6284.
14. Creating Chemical Diversity Space by Scaffold Decoration of Dihydropyrimidines.
D. Dallinger, C.O. Kappe
Pure Appl. Chem. 2005, 77, 155-161.
15. The Impact of Microwave Synthesis on Drug Discovery.
C.O. Kappe, D. Dallinger
Nature Rev. Drug. Discov. 2006, 5, 51-63.
16. The Use of Microwave Irradiation in Organic Synthesis. From Laboratory Curiosity to Standard Practice in Twenty Years.
C.O. Kappe
Chimia 2006, 60, 308-312.
17. Microwave-Assisted Synthesis under Continuous Flow Conditions.
T. N. Glasnov, C.O. Kappe
Macromol. Rapid Commun. 2007, 28, 395-410.
18. Microwave Synthesis in High-Throughput Environments. Moving from Automated Sequential to Microtiter Plate Formats.
M. Matloobi, C.O. Kappe
Chim. Oggi 2007, 25, 26-31.
19. Microwave-Assisted Synthesis in Water as Solvent.
D. Dallinger, C.O. Kappe
Chem. Rev. 2007, 107, 2563-2591.
20. Parallel Processing of Microwave-Assisted Organic Transformations.
M. Matloobi, C.O. Kappe
Comb. Chem. High Throughp. Screening 2007, 10, 735-750.
21. Copper-Catalyzed C-C Coupling of Thiol Esters and Boronic Acids under Aerobic Conditions.
H. Prokopcova, C.O. Kappe
Angew. Chem. Int. Ed. 2008, 47, 3674-3677.
22. Microwave Dielectric Heating in Synthetic Organic Chemistry.
C.O. Kappe
Chem. Sov. Rev. 2008, 37, 1127-1139.
23. The Liebeskind-Srogl C-C Cross-Coupling Reaction.
H. Prokopcova, C.O. Kappe
Angew. Chem. Int. Ed. 2009, 48, 2276.
24. Controlled Microwave Heating in Modern Organic Synthesis. Highlights from the 2004-2008 Literature.
C. O. Kappe, D. Dallinger
Mol. Diversity 2009, 13, 71-193.
25. Click Chemistry under Non-classical Reaction Conditions.
C.O. Kappe, E. Van der Eycken
Chem. Sov. Rev. 2010, 39, 1280-1290.
26. Heterocyclic BINAP Analogues.
N. Arshad, C. O. Kappe
Adv. Heterocycl. Chem. 2010, 99, 33-59.
27. Continuous Flow Organic Synthesis Under High Temperature/Pressure Conditions.
T. Razzaq, C.O. Kappe
Chem. Asian J. 2010, 5, 1274-1289.
28. Microwave-assisted Derivatization Procedures for Gas Chromatography/Mass Spectrometry Analysis.
S. L. Söderholm, M. Damm, C. O. Kappe
Mol. Diversity 2010, 14, 869-868.
29. Continuous Flow Synthesis of Heterocycles.
T. N. Glasnov, C. O. Kappe
J. Heterocycl. Chem. 2011, 48, 11-29.
30. Heterogeneous Catalytic Hydrogenation Reactions Using Continuous Flow Reactors.
M. Irfan, T. N. Glasnov, C. O. Kappe
ChemSusChem, 2011, 4, 300-316.
31. A Critical Assessment of the Greenness and Energy Efficiency of Microwave-assisted Organic Synthesis.
J. D. Moseley, C. O. Kappe
Green Chem. 2011, 13, 794-806.
32. The Microwave-to-Flow Paradigm: Translating High-Temperature Batch Microwave Chemistry to Scalable Continuous Flow Processes.
T. N. Glasnov, C. O. Kappe
Chem. Eur. J. 2011, 17, 11956-11968.
33. Microwave-Assisted Synthesis of Colloidal Inorganic Nanocrystals.
M. Baghbanzadeh, L. Carbone, P. D. Cozzoli, C. O. Kappe
Angew. Chem. Int. Ed. 2011, 50, 11312-11359.
34. Parallel Microwave Chemistry in Silicon Carbide Microtiter Platforms – A Review
C. O. Kappe, M. Damm
Mol. Diversity 2012, 16, 5-25.
